ASF1A-dependent P300-mediated histone H3 lysine 18 lactylation promotes atherosclerosis by regulating EndMT

ASF1A-dependent P300-mediated histone H3 lysine 18 lactylation promotes atherosclerosis by regulating EndMT

2024 | Mengdie Dong, Yunjia Zhang, Minghong Chen, Yongkang Tan, Jiao Min, Xian He, Fuhao Liu, Jiaming Gu, Hong Jiang, Longbin Zheng, Jiajing Chen, Quanwen Yin, Xuesong Li, Xiang Chen, Yongfeng Shao, Yong Ji, Hongshan Chen
Atherosclerosis is a chronic inflammatory vascular disease driven by endothelial-to-mesenchymal transition (EndMT). This study reveals that lipid peroxidation promotes EndMT by increasing lactate-dependent histone H3 lysine 18 lactylation (H3K18la). The histone chaperone ASF1A, identified as a cofactor of P300, precisely regulates H3K18la at the SNAI1 promoter, activating SNAI1 transcription and promoting EndMT. ASF1A deletion inhibits EndMT and improves endothelial dysfunction. In atherosclerosis models, endothelium-specific ASF1A deficiency reduces EndMT and alleviates atherosclerosis. Pharmacological inhibition of glycolysis and PROTACs reduce H3K18la, SNAI1 transcription, and EndMT-induced atherosclerosis. The study highlights the crosstalk between metabolism and epigenetics via H3K18la mediated by the P300/ASF1A complex during EndMT, offering new therapeutic strategies for atherosclerosis.Atherosclerosis is a chronic inflammatory vascular disease driven by endothelial-to-mesenchymal transition (EndMT). This study reveals that lipid peroxidation promotes EndMT by increasing lactate-dependent histone H3 lysine 18 lactylation (H3K18la). The histone chaperone ASF1A, identified as a cofactor of P300, precisely regulates H3K18la at the SNAI1 promoter, activating SNAI1 transcription and promoting EndMT. ASF1A deletion inhibits EndMT and improves endothelial dysfunction. In atherosclerosis models, endothelium-specific ASF1A deficiency reduces EndMT and alleviates atherosclerosis. Pharmacological inhibition of glycolysis and PROTACs reduce H3K18la, SNAI1 transcription, and EndMT-induced atherosclerosis. The study highlights the crosstalk between metabolism and epigenetics via H3K18la mediated by the P300/ASF1A complex during EndMT, offering new therapeutic strategies for atherosclerosis.
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