Lactylated Apolipoprotein C-II Induces Immunotherapy Resistance by Promoting Extracellular Lipolysis

Lactylated Apolipoprotein C-II Induces Immunotherapy Resistance by Promoting Extracellular Lipolysis

2024 | Jian Chen, Deping Zhao, Yupeng Wang, Ming Liu, Yuan Zhang, Tingting Feng, Chao Xiao, Huan Song, Rui Miao, Li Xu, Hongwei Chen, Xiaoying Qiu, Yi Xu, Jingxuan Xu, Zelin Cui, Wei Wang, Yanchun Quan, Yifeng Zhu, Chen Huang, Song Guo Zheng, Jian-yuan Zhao, Ting Zhu, Lianhui Sun, Guangjian Fan
Lactylated apolipoprotein C-II (APOC2) promotes extracellular lipolysis, leading to immunotherapy resistance in non-small-cell lung cancer (NSCLC). This study reveals that lactate induces lactyl-APOC2-K70, which stabilizes APOC2 and increases free fatty acid (FFA) release, promoting regulatory T cell (Treg) accumulation and tumor metastasis. Mechanistically, lactate enhances APOC2 lactylation at K70, stabilizing the protein and facilitating FFA release. This process is mediated by P300, which promotes APOC2-K70 lactylation, while HDAC3 delactylates APOC2. The anti-APOC2-K70-lac antibody sensitizes anti-PD-1 therapy by inhibiting lactyl-APOC2, reducing Treg accumulation and enhancing immunotherapy efficacy. Lactyl-APOC2-K70 is associated with tumor progression and immunotherapy resistance in NSCLC samples, with higher levels correlating with poor prognosis. The findings highlight the potential of targeting lactyl-APOC2-K70 as a novel therapeutic strategy for NSCLC.Lactylated apolipoprotein C-II (APOC2) promotes extracellular lipolysis, leading to immunotherapy resistance in non-small-cell lung cancer (NSCLC). This study reveals that lactate induces lactyl-APOC2-K70, which stabilizes APOC2 and increases free fatty acid (FFA) release, promoting regulatory T cell (Treg) accumulation and tumor metastasis. Mechanistically, lactate enhances APOC2 lactylation at K70, stabilizing the protein and facilitating FFA release. This process is mediated by P300, which promotes APOC2-K70 lactylation, while HDAC3 delactylates APOC2. The anti-APOC2-K70-lac antibody sensitizes anti-PD-1 therapy by inhibiting lactyl-APOC2, reducing Treg accumulation and enhancing immunotherapy efficacy. Lactyl-APOC2-K70 is associated with tumor progression and immunotherapy resistance in NSCLC samples, with higher levels correlating with poor prognosis. The findings highlight the potential of targeting lactyl-APOC2-K70 as a novel therapeutic strategy for NSCLC.
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